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Breadcrumb Research A-Z researchers William McCarthy Postdoctoral Fellow Rittinger lab Molecular Structure of Cell Signalling Laboratory Email Address: Email Year published 2026 (1) 2025 (2) 2024 (1) 2023 (2) Facet Year published Research topics Biochemistry & Proteomics (2) Chemical Biology & High Throughput (6) Computational & Systems Biology (2) Genetics & Genomics (2) Infectious Disease (3) Structural Biology & Biophysics (1) Facet Research topics Crick Pre-Crick Crick publications (6) Facet Crick Pre-Crick Publication type Journal article (6) Primary research (5) Review (1) Facet Publication type Journal Angewandte Chemie (1) Angewandte Chemie International Edition (1) Communications Chemistry (1) Current Opinion in Structural Biology (1) Nature Communications (1) RSC Chemical Biology (1) Facet Journal Displaying 1 - 6 of 6Last updated : 03 March 2026 03:05 Covalent fragment screening to inhibit the E3 ligase activity of bacterial NEL enzymes SspH1 and SspH2 Authors (12) Cassandra Kennedy Katherine McPhie Aini Vuorinen Jane Dudley Diego Esposito Sarah Maslen [...] Jonathan Pettinger Mark Skehel Jacob Bush David House Katrin Rittinger RSC Chemical Biology Published 1 January 2026 Crick labs/ facilities Katrin Rittinger Proteomics Full details Enantioselective OTUD7B fragment discovery through chemoproteomics screening and high-throughput optimisation Authors (9) Aini Vuorinen Cassandra Kennedy Katherine McPhie William McCarthy Jonathan Pettinger Mark Skehel David House Jacob T Bush Katrin Rittinger Communications Chemistry Published 15 January 2025 Crick labs/ facilities Katrin Rittinger Proteomics Scientific computing Cell Science Full details Robust proteome profiling of cysteine-reactive fragments using label-free chemoproteomics Authors (16) George S Biggs Emma Cawood Aini Vuorinen William McCarthy Harry Wilders Ioannis G Riziotis [...] David House Simon Boulton Mark Skehel Katrin Rittinger Jacob T Bush Nature Communications Published 2 January 2025 Crick labs/ facilities Katrin Rittinger Simon Boulton Scientific computing Proteomics Cell Science Full details Covalent fragment-based drug discovery for target tractability Authors (4) William McCarthy Niek vanderZouwen Jacob T Bush Katrin Rittinger Current Opinion in Structural Biology Published 1 June 2024 Crick labs Katrin Rittinger Full details Chemical validation of Mycobacterium tuberculosis phosphopantetheine adenylyltransferase using fragment linking and CRISPR interference Authors (13) Jamal El Bakali Michal Blaszczyk Joanna Evans Jennifer A Boland William McCarthy Imam Fathoni [...] Anthony G Coyne Valerie Mizrahi Tom L Blundell Chris Abell Christina Spry Angewandte Chemie International Edition Published 17 April 2023 Crick labs Eachan Johnson Full details Chemical validation of Mycobacterium tuberculosis phosphopantetheine adenylyltransferase using fragment linking and CRISPR interference Authors (13) Jamal El Bakali Michal Blaszczyk Joanna Evans Jennifer A Boland William McCarthy Imam Fathoni [...] Anthony G Coyne Valerie Mizrahi Tom L Blundell Chris Abell Christina Spry Angewandte Chemie Published 17 April 2023 Crick labs Eachan Johnson Full details
Covalent fragment screening to inhibit the E3 ligase activity of bacterial NEL enzymes SspH1 and SspH2 Authors (12) Cassandra Kennedy Katherine McPhie Aini Vuorinen Jane Dudley Diego Esposito Sarah Maslen [...] Jonathan Pettinger Mark Skehel Jacob Bush David House Katrin Rittinger RSC Chemical Biology Published 1 January 2026 Crick labs/ facilities Katrin Rittinger Proteomics Full details
Enantioselective OTUD7B fragment discovery through chemoproteomics screening and high-throughput optimisation Authors (9) Aini Vuorinen Cassandra Kennedy Katherine McPhie William McCarthy Jonathan Pettinger Mark Skehel David House Jacob T Bush Katrin Rittinger Communications Chemistry Published 15 January 2025 Crick labs/ facilities Katrin Rittinger Proteomics Scientific computing Cell Science Full details
Robust proteome profiling of cysteine-reactive fragments using label-free chemoproteomics Authors (16) George S Biggs Emma Cawood Aini Vuorinen William McCarthy Harry Wilders Ioannis G Riziotis [...] David House Simon Boulton Mark Skehel Katrin Rittinger Jacob T Bush Nature Communications Published 2 January 2025 Crick labs/ facilities Katrin Rittinger Simon Boulton Scientific computing Proteomics Cell Science Full details
Covalent fragment-based drug discovery for target tractability Authors (4) William McCarthy Niek vanderZouwen Jacob T Bush Katrin Rittinger Current Opinion in Structural Biology Published 1 June 2024 Crick labs Katrin Rittinger Full details
Chemical validation of Mycobacterium tuberculosis phosphopantetheine adenylyltransferase using fragment linking and CRISPR interference Authors (13) Jamal El Bakali Michal Blaszczyk Joanna Evans Jennifer A Boland William McCarthy Imam Fathoni [...] Anthony G Coyne Valerie Mizrahi Tom L Blundell Chris Abell Christina Spry Angewandte Chemie International Edition Published 17 April 2023 Crick labs Eachan Johnson Full details
Chemical validation of Mycobacterium tuberculosis phosphopantetheine adenylyltransferase using fragment linking and CRISPR interference Authors (13) Jamal El Bakali Michal Blaszczyk Joanna Evans Jennifer A Boland William McCarthy Imam Fathoni [...] Anthony G Coyne Valerie Mizrahi Tom L Blundell Chris Abell Christina Spry Angewandte Chemie Published 17 April 2023 Crick labs Eachan Johnson Full details